2
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP2160L1 | YAP-TEAD-IN-1 acetate | YAP-TEAD-IN-1 acetate (1659305-78-8 Free base) | YAP |
YAP-TEAD-IN-1 acetate is an effective and competitive inhibitor of YAP–TEAD interaction with an IC50 of 25 nM. | |||
TP2160 | YAP-TEAD-IN-1 | Others | |
YAP-TEAD-IN-1 is a competitive inhibitor of YAP–TEAD interaction (IC50: 25 nM). It shows a higher binding affinity to TEAD1 (Kd: 15 nM) than YAP (50-171) (Kd: 40 nM). |